3D QSAR study, synthesis, and in vitro evaluation of (+)-5-FBVM as potential PET radioligand for the vesicular acetylcholine transporter (VAChT)

Sylvie Mavel (1) , Mitja Kovac , Winnie Deuther-Conrad (2) , Nathalie Méheux , Jana Glöckner , Barbara Wenzel (2) , Marko Anderluh (3) , Peter Brust (2) , Denis Guilloteau (4) , Patrick Emond (4)

1 Equipe neurogénétique et neurométabolomique
2 Institute of Radiopharmaceutical Cancer Research
3 inconnu
4 iBrain - Inserm U1253 - UNIV Tours - Imagerie et cerveau

Domains: Chemical Sciences; Medicinal Chemistry

Sylvie Mavel, Mitja Kovac, Winnie Deuther-Conrad, Nathalie Méheux, Jana Glöckner, et al.. 3D QSAR study, synthesis, and in vitro evaluation of (+)-5-FBVM as potential PET radioligand for the vesicular acetylcholine transporter (VAChT). Bioorganic and Medicinal Chemistry, 2010, 18 (21), pp.7659 - 7667. ⟨10.1016/j.bmc.2010.08.028⟩. ⟨hal-01826409⟩